Empesertib (BAY 1161909)

CAS No. 1443763-60-7

Empesertib (BAY 1161909)( BAY 1161909 )

Catalog No. M21766 CAS No. 1443763-60-7

BAY 1161909 is a potent Mps1 inhibitor, with an IC50 of < 1 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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2MG 176 In Stock
5MG 290 In Stock
10MG 435 In Stock
25MG 710 In Stock
50MG 972 In Stock
100MG 1341 In Stock
500MG 2682 In Stock
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Biological Information

  • Product Name
    Empesertib (BAY 1161909)
  • Note
    Research use only, not for human use.
  • Brief Description
    BAY 1161909 is a potent Mps1 inhibitor, with an IC50 of < 1 nM.
  • Description
    BAY 1161909 is a potent Mps1 inhibitor, with an IC50 of < 1 nM. BAY 1161909 also shows anti-tumor effect, suppressing the proliferation of Hela cells, with an IC50 of < 400 nM.(In Vitro):BAY 1161909 is a potent Mps1 inhibitor, with an IC50 of < 1 nM. BAY 1161909 also shows anti-tumor effect, suppressing the proliferation of Hela cells, with an IC50 of < 400 nM.
  • In Vitro
    BAY 1161909 is a potent Mps1 inhibitor, with an IC50 of < 1 nM. BAY 1161909 also shows anti-tumor effect, suppressing the proliferation of Hela cells, with an IC50 of < 400 nM.
  • In Vivo
    ——
  • Synonyms
    BAY 1161909
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    Mps1/TTK
  • Recptor
    ——
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1443763-60-7
  • Formula Weight
    559.61
  • Molecular Formula
    C??H??FN?O?S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO : ≥ 35 mg/mL (62.54 mM) H2O : < 0.1 mg/mL (insoluble)
  • SMILES
    FC1=CC=C([C@@H](C)C(NC2=CC=C(C3=CN4N=C(NC5=CC=C(S(C)(=O)=O)C=C5OC)N=C4C=C3)C=C2)=O)C=C1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. SCHULZE, Volker, et al. PRODRUG DERIVATIVES OF SUBSTITUTED TRIAZOLOPYRIDINES. WO2014198647A2
molnova catalog
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    BAY 1161909 is a potent Mps1 inhibitor, with an IC50 of < 1 nM.