
Empesertib (BAY 1161909)
CAS No. 1443763-60-7
Empesertib (BAY 1161909)( BAY 1161909 )
Catalog No. M21766 CAS No. 1443763-60-7
BAY 1161909 is a potent Mps1 inhibitor, with an IC50 of < 1 nM.
Purity : >98% (HPLC)






Size | Price / USD | Stock | Quantity |
2MG | 176 | In Stock |
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5MG | 290 | In Stock |
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10MG | 435 | In Stock |
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25MG | 710 | In Stock |
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50MG | 972 | In Stock |
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100MG | 1341 | In Stock |
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500MG | 2682 | In Stock |
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1G | Get Quote | In Stock |
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Biological Information
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Product NameEmpesertib (BAY 1161909)
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NoteResearch use only, not for human use.
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Brief DescriptionBAY 1161909 is a potent Mps1 inhibitor, with an IC50 of < 1 nM.
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DescriptionBAY 1161909 is a potent Mps1 inhibitor, with an IC50 of < 1 nM. BAY 1161909 also shows anti-tumor effect, suppressing the proliferation of Hela cells, with an IC50 of < 400 nM.(In Vitro):BAY 1161909 is a potent Mps1 inhibitor, with an IC50 of < 1 nM. BAY 1161909 also shows anti-tumor effect, suppressing the proliferation of Hela cells, with an IC50 of < 400 nM.
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In VitroBAY 1161909 is a potent Mps1 inhibitor, with an IC50 of < 1 nM. BAY 1161909 also shows anti-tumor effect, suppressing the proliferation of Hela cells, with an IC50 of < 400 nM.
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In Vivo——
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SynonymsBAY 1161909
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PathwayCell Cycle/DNA Damage
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TargetMps1/TTK
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number1443763-60-7
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Formula Weight559.61
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Molecular FormulaC??H??FN?O?S
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Purity>98% (HPLC)
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SolubilityDMSO : ≥ 35 mg/mL (62.54 mM) H2O : < 0.1 mg/mL (insoluble)
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SMILESFC1=CC=C([C@@H](C)C(NC2=CC=C(C3=CN4N=C(NC5=CC=C(S(C)(=O)=O)C=C5OC)N=C4C=C3)C=C2)=O)C=C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. SCHULZE, Volker, et al. PRODRUG DERIVATIVES OF SUBSTITUTED TRIAZOLOPYRIDINES. WO2014198647A2
molnova catalog



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Empesertib (BAY 1161...
BAY 1161909 is a potent Mps1 inhibitor, with an IC50 of < 1 nM.